Development

Apogee Therapeutics' zumilokibart maintains atopic dermatitis responses with every-three-to-six-month dosing in Phase II trial

Apogee Therapeutics (Nasdaq: APGE), a clinical-stage biotech based in San Francisco and Boston, reported 52-week maintenance data from the Phase II APEX Part A trial of zumilokibart (APG777) in moderate-to-severe atopic dermatitis, with results showing that patients maintained and deepened clinical responses on dosing schedules of every three or six months. If confirmed in placebo-controlled and Phase III studies, the zumilokibart atopic dermatitis data could position the anti-IL-13 antibody as a less frequently dosed alternative to current biologics that require injections as often as every two weeks.

The APEX trial (NCT05942655) is a Phase II study evaluating zumilokibart at 360mg administered subcutaneously at three- and six-month intervals in adults with moderate-to-severe atopic dermatitis. Part A assessed maintenance of response over 52 weeks among patients who had completed a 16-week induction period.

Zumilokibart Phase 2 Results: Maintenance and Deepening of Responses

Among patients who achieved response at Week 16, 75% and 85% maintained EASI-75 — a 75% or greater reduction in the Eczema Area and Severity Index — with every three-month and every six-month dosing, respectively. Maintenance of clear or almost clear skin, measured by validated Investigator's Global Assessment (vIGA) scores of 0 or 1, was observed in 86% of patients on three-month dosing and 78% on six-month dosing. The company also reported that deepening of response occurred across all lesional and itch endpoints in the full population of patients initially randomized to zumilokibart, not solely among Week 16 responders. The EASI-75 zumilokibart results, together with the vIGA data, form the core of the efficacy case the company is building ahead of Phase III.

Zumilokibart was well tolerated across both dosing regimens over the full 52-week study period. The most common treatment-emergent adverse events were noninfective conjunctivitis, upper respiratory tract infection, and nasopharyngitis — a profile the company described as generally consistent with other agents in the IL-13 inhibitor class.

Mechanism and Drug Context: How APG777 Targets IL-13

Zumilokibart is a subcutaneous monoclonal antibody engineered with an extended half-life that targets interleukin-13, a cytokine considered a primary driver of the inflammation, barrier dysfunction, and pruritus characteristic of atopic dermatitis. According to the company, zumilokibart achieves greater than 99% inhibition of IL-13, which Apogee Therapeutics argues underpins the rapid onset and sustained depth of response observed in the APEX trial atopic dermatitis data. The extended half-life engineering is what enables the three- and six-month dosing intervals that distinguish the Apogee Therapeutics APG777 program from existing biologics in the class.

Positioning Among Current Moderate-to-Severe Atopic Dermatitis Treatments

The moderate-to-severe atopic dermatitis treatment landscape has expanded in recent years with the approval of dupilumab (Dupixent), an anti-IL-4 receptor alpha antibody administered every two weeks; tralokinumab (Adbry), an anti-IL-13 antibody dosed every two weeks during induction and every two to four weeks thereafter; and oral JAK inhibitors including upadacitinib (Rinvoq) and abrocitinib (Cibinqo). Dupilumab remains the most widely prescribed biologic in the indication.

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Tralokinumab is the most direct comparator for zumilokibart given their shared IL-13 target. In its pivotal trials, tralokinumab demonstrated EASI-75 rates of approximately 25–33% at Week 16 versus placebo rates of around 10–13%, with maintenance dosing every two weeks or every four weeks. The zumilokibart maintenance data — showing 75–85% of Week 16 responders maintaining EASI-75 at 52 weeks on three- or six-month dosing — appear numerically distinct in terms of dosing frequency, though cross-trial comparisons are limited by differences in study design, patient populations, and the absence of a placebo arm in the APEX Part A maintenance phase. The Part A data represent a responder-enriched population, which inflates absolute response rates relative to intent-to-treat analyses from pivotal trials.

The dosing interval is the central differentiator. Current standard-of-care biologics require between 13 and 26 injections per year. If zumilokibart's efficacy and safety are confirmed in controlled studies, a regimen of two to four doses per year would represent a meaningful reduction in treatment burden. Whether this translates into improved adherence and real-world outcomes remains to be determined.

What Comes Next for the APEX Trial and Zumilokibart Development

APEX Part B, a placebo-controlled dose optimization segment that randomized 347 patients 1:1:1:1 to high-, medium-, or low-dose zumilokibart versus placebo, is expected to report 16-week induction data in the second quarter of 2026. That readout will provide the first controlled efficacy comparison for the molecule in atopic dermatitis and will be a more informative test of zumilokibart's treatment effect size relative to placebo.

Based on the Part A and anticipated Part B results, Apogee plans to initiate Phase III trials of zumilokibart in moderate-to-severe atopic dermatitis in the second half of 2026, with a potential commercial launch targeted for 2029. The 52-week data will be presented in a late-breaking oral presentation at the 2026 American Academy of Dermatology Annual Meeting on March 28 in Denver.

The company has also disclosed plans to expand zumilokibart's development into asthma, eosinophilic esophagitis, and other inflammatory and immunology indications, though timelines for those programs were not specified in the current disclosure.


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