Development

Cytokinetics' aficamten meets endpoints in Phase III non-obstructive cardiomyopathy trial, nudging ahead of BMS

Cytokinetics (Nasdaq: CYTK) reported that aficamten met both dual primary endpoints in the Phase III ACACIA-HCM trial in symptomatic non-obstructive hypertrophic cardiomyopathy, a patient population for which no disease-specific therapy is currently approved by the FDA or EMA. The aficamten hypertrophic cardiomyopathy data, drawn from 516 randomized participants, showed statistically significant improvements in both symptom burden and exercise capacity compared to placebo at 36 weeks — the first Phase III trial to demonstrate such improvements in this subtype.

ACACIA-HCM Trial Results: What the Data Show

The ACACIA-HCM trial is a Phase III, multi-center, randomized, double-blind, placebo-controlled study designed to evaluate aficamten against placebo in adults with symptomatic non-obstructive HCM, enrolling 516 participants outside Japan on a 1:1 basis.

On the dual primary endpoints, aficamten produced a least square mean change in Kansas City Cardiomyopathy Questionnaire Clinical Summary Score (KCCQ-CSS) of 11.4 points from baseline versus 8.4 points for placebo, a treatment difference of 3.0 points (95% CI: 0.5–5.5; p=0.021). The KCCQ cardiac outcomes signal was consistent throughout the treatment period and reversed toward placebo levels following washout, suggesting an on-target pharmacological effect rather than a sustained structural change. On maximal exercise performance, peak oxygen consumption (pVO2) increased by 0.64 mL/kg/min with aficamten versus a decline of 0.03 mL/kg/min with placebo, a difference of 0.67 mL/kg/min (95% CI: 0.22–1.1; p=0.003).

Key secondary endpoints, each reaching p<0.001, included the proportion of participants achieving at least one class improvement in New York Heart Association functional class, a composite z-score of ventilatory efficiency and pVO2, and NT-proBNP reduction. The consistency of these findings across both patient-reported and physician-assessed measures strengthens the overall signal, though the magnitude of the KCCQ difference — 3.0 points — sits at the lower boundary of what is generally considered clinically meaningful in cardiomyopathy trials, a nuance that regulators are likely to weigh carefully.

Safety profile

No new safety signals were identified. Completion of planned dosing was similar between arms: 88.4% for aficamten and 90.3% for placebo. However, the reduction in left ventricular ejection fraction (LVEF) below 50% occurred in 10% of aficamten-treated participants compared to 1% on placebo, and two participants on aficamten experienced serious adverse events of heart failure associated with that LVEF decline. Treatment interruptions due to LVEF falling below 40% occurred in 3% of the aficamten group.

This safety pattern is consistent with the known pharmacology of cardiac myosin inhibitors and mirrors the profile established in obstructive HCM trials. Myqorzo (aficamten), already approved in the US, EU, and China for symptomatic obstructive HCM, carries a boxed warning for the risk of heart failure due to systolic dysfunction and is available only through a Risk Evaluation and Mitigation Strategy (REMS) program in the US.

The competitive context for aficamten in hypertrophic cardiomyopathy

Non-obstructive HCM accounts for approximately half of all HCM cases based on recent claims data analysis, representing an estimated 150,000 or more diagnosed patients in the US alone. Unlike obstructive HCM, where the left ventricular outflow tract gradient provides both a pathophysiological target and a measurable surrogate endpoint, non-obstructive disease is defined by the absence of that gradient — meaning the disease burden falls almost entirely on symptoms, diastolic dysfunction, and exercise intolerance, with no pharmacological intervention currently holding regulatory approval.

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Cytokinetics aficamten program is the first to generate Phase III evidence in this setting. Bristol Myers Squibb's Camzyos (mavacamten), the first cardiac myosin inhibitor to reach market, was approved by the FDA in April 2022 for symptomatic obstructive HCM. BMS has not reported pivotal Phase III data in non-obstructive HCM, making the ACACIA-HCM trial results the first positive Phase III dataset in that subtype from either agent in the class. Cross-trial comparisons between aficamten and mavacamten are limited by differences in trial design, patient populations, and endpoint definitions, but the non-obstructive indication represents potential commercial and clinical differentiation for Cytokinetics if regulatory approval follows.

Aficamten was engineered to achieve a more predictable exposure-response relationship than mavacamten, with dose titration guided by echocardiographic LVEF monitoring at weeks 2, 4, and 6. In ACACIA-HCM, participants began at 5 mg once daily and could be escalated to 10, 15, or 20 mg provided LVEF remained at or above 60%. That titration framework mirrors the approach used in obstructive HCM trials and is intended to manage the systolic dysfunction risk inherent to the mechanism.

What Comes Next for the Cytokinetics Aficamten Program

Cytokinetics stated it plans to present full ACACIA-HCM trial results at an upcoming medical meeting and to discuss the data with the FDA and other regulatory authorities. The company has not yet announced a submission timeline for a non-obstructive HCM indication. Aficamten is also under investigation in CEDAR-HCM, a pediatric study in obstructive HCM, and in FOREST-HCM, an open-label extension study, though neither of those programs bears directly on the non-obstructive adult indication under review here.

The regulatory path for the non-obstructive indication will likely require scrutiny of the absolute KCCQ treatment difference and the LVEF safety data, particularly given that the non-obstructive population has no established pharmacological comparator against which to contextualize benefit-risk. Full data disclosure at a major cardiology meeting will be the next material event for investors and clinicians tracking this program.


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