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Amgen/AZ's Tezspire extends TSLP platform to eosinophilic esophagitis with Phase III win

Amgen/AZ's Tezspire extends TSLP platform to eosinophilic esophagitis with Phase III win

Tezepelumab has met both co-primary and all key secondary endpoints in eosinophilic esophagitis, Amgen (Nasdaq: AMGN) and AstraZeneca reported on August 27, extending the anti-thymic stromal lymphopoietin (TSLP) antibody's demonstrated efficacy to a third epithelial-driven inflammatory disease after severe asthma and chronic rhinosinusitis with nasal polyps (CRSwNP).

The Phase III CROSSING trial enrolled 368 patients aged 12–80 years with symptomatic, histologically active eosinophilic esophagitis (EoE) uncontrolled on maintenance therapy, randomized 1:1:1 to low-dose tezepelumab, high-dose tezepelumab, or placebo, all administered subcutaneously every four weeks. Co-primary endpoints at week 24 were histologic remission — defined as a peak esophageal eosinophil count of six or fewer per high-power field — and mean change from baseline in the patient-reported Dysphagia Symptom Questionnaire (DSQ) score. Both were met with statistically significant and clinically meaningful improvements versus placebo, the companies said, and those improvements were sustained through week 52. All key secondary endpoints, including endoscopic disease features, histologic severity, and total endoscopic remission at week 52, were also met. Specific numerical results have not been disclosed; full data will be presented at an upcoming medical meeting.

The safety profile was described as generally consistent with tezepelumab's approved indications. Tezepelumab (Tezspire) is currently approved for severe asthma in the US, EU, China, Japan, and more than 70 countries, and received FDA approval for CRSwNP in October 2025 based on the Phase III WAYPOINT trial, which showed a 98% reduction in surgery need and 88% reduction in systemic corticosteroid use versus placebo.

Tezepelumab blocks TSLP, an epithelial cytokine that sits upstream of multiple inflammatory cascades. In EoE, TSLP is preferentially secreted by terminally differentiated esophageal epithelial cells and is believed to initiate the eosinophilic inflammation that drives dysphagia, food impaction, and esophageal remodeling. By acting at this upstream checkpoint rather than targeting downstream mediators such as IL-5 or IL-13, tezepelumab intervenes earlier in the inflammatory cascade rather than targeting individual effector pathways — a distinction the companies have consistently emphasized across indications.

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The EoE market currently has one approved biologic: Sanofi and Regeneron's Dupixent (dupilumab), which blocks IL-4 receptor alpha signaling and was first approved by the FDA for EoE in May 2022, with a pediatric expansion to children aged one year and older in January 2024. Takeda's Eohilia (budesonide oral suspension) received FDA approval in February 2024 as the first oral pharmacotherapy for EoE, though it is indicated only for a 12-week course rather than chronic maintenance. Bristol Myers Squibb's cendakimab, an anti-IL-13 antibody that completed a positive Phase III trial in EoE, was discontinued in February 2025 as part of pipeline cost-cutting. Tezepelumab's upstream TSLP mechanism differentiates it from the approved and discontinued agents, which target downstream type 2 cytokines; whether that translates to a clinical advantage over dupilumab will require head-to-head data that do not yet exist.

For Amgen and AstraZeneca, a positive EoE filing would extend tezepelumab's label across three distinct epithelial-driven conditions and reinforce the commercial and scientific rationale for the TSLP platform. The drug also holds FDA Orphan Drug Designation for EoE, granted in October 2021. Phase III COPD trials — JOURNEY and EMBARK — are ongoing, and the FDA granted a Breakthrough Therapy Designation for tezepelumab in eosinophilic COPD in July 2024, meaning EoE would represent one of potentially four approved indications if both programs succeed. The companies said they will submit the CROSSING data to regulatory authorities as quickly as possible.


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