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Ten63 Therapeutics Closes Strategic Financing Round Bringing Total Funding Past USD 45 Million

Ten63 Therapeutics, a Durham, North Carolina–based AI drug discovery company developing small molecules against targets long considered undruggable, has...

Ten63 Therapeutics Closes Strategic Financing, Bringing Total Funding Past USD 45m

Ten63 Therapeutics, a Durham, North Carolina–based AI drug discovery company developing small molecules against targets long considered undruggable, has closed a strategic financing round that brings its total funding to more than USD 45 million. The company, which is built around a proprietary computational platform called BEYOND, did not disclose the specific amount raised in this latest tranche. Ten63 said the capital will be used to scale its AI-driven drug discovery platform and advance an internal oncology pipeline focused on targets that have resisted decades of conventional drug development efforts.

Chugai Venture Fund, Gates Foundation Among New Backers

The round drew new investment from Chugai Venture Fund — the venture arm of Japanese pharmaceutical company Chugai Pharmaceutical Co., Ltd. — and the Bill & Melinda Gates Foundation. Additional new investors included RYSE, K5 Global, SF Holdings, Duke Capital Partners, Cape Fear BioCapital, Black Opal Ventures, and Panorama. They joined an existing syndicate comprising Hatteras Venture Partners, Yosemite, Morpheus Ventures, Alexandria Venture Investments, and Draper Associates, the company said.

In connection with the financing, Mike Dial, Ph.D., Managing Director of Chugai Venture Fund, joined Ten63's board of directors.

The company said the increased funding will fuel further development of the BEYOND discovery platform and support the advancement of its preclinical pipeline. Ten63 also received a grant from the Gates Foundation — separate from the equity investment — to support work on affordable small-molecule therapeutics targeting human papillomavirus (HPV), the most common sexually transmitted infection worldwide and a leading cause of cervical cancer.

Preclinical Pipeline Targets Myc and HPV Viral Proteins

Ten63 does not appear to have any active clinical-stage programs registered in public trial databases. The company's pipeline is preclinical and centers on what it describes as first- and best-in-class small molecules against oncology targets that have historically been considered undruggable.

The most prominently discussed program targets Myc, an oncogene implicated in an estimated 70% of all cancers. Myc has been a subject of drug discovery efforts for more than four decades, but no approved therapy directly inhibits the protein. Ten63 said it has Myc-targeting therapeutics in active preclinical development that it claims surpass all previous attempts at Myc inhibition, though no peer-reviewed data supporting this assertion have been publicly disclosed.

A second disclosed area of focus involves HPV-associated cancers. HPV causes cancer in more than 650,000 women and men each year globally, and while vaccines exist for prevention, treatment options for established HPV lesions — particularly in low- and middle-income countries — remain limited. Ten63 said its BEYOND platform is being applied to develop cost-effective small molecules targeting viral proteins that drive HPV-related malignancies. This work is being conducted with support from the Gates Foundation grant and in collaboration with researchers at the University of Oxford.

External sources have also indicated that Ten63 has a KRAS G12D inhibitor at the preclinical stage for neoplasms, though the company did not reference this program in its latest announcement.

The BEYOND Platform: Large Quantum Chemistry Models for Artificial Intelligence Drug Discovery

The BEYOND platform — which stands for Binding Evolution Yields Original New Drugs — is described by Ten63 as the world's first Large Quantum Chemistry Model (LQCM). The company says the platform delivers quantum-mechanics-level simulations at speeds orders of magnitude faster than other computational approaches, enabling it to simulate trillions of potential drug molecules per protein target while retaining accuracy approaching that of laboratory experiments.

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The scientific rationale underpinning the platform addresses a well-documented constraint in drug discovery: approximately 80% of all human proteins lack the well-defined binding pockets that conventional small-molecule screening depends on. These so-called undruggable targets include transcription factors like Myc and certain viral proteins. Traditional high-throughput screening and structure-based drug design have largely failed against such targets because they present shallow, transient, or poorly characterized interaction surfaces.

Ten63 contends that BEYOND overcomes these limitations by using AI to explore chemical space computationally at a scale and resolution that physical screening cannot match. The platform generates and evaluates molecular candidates through iterative cycles that the company likens to evolutionary selection, optimizing for binding, selectivity, and drug-like properties against targets where conventional methods have not produced viable candidates.

Marcel Frenkel, Ph.D., CEO of Ten63, said in a statement that the platform is "advancing towards superintelligence for drug discovery," adding that "at that point, we believe little will remain undruggable." John Gustofson, President and Head of Chugai Venture Fund, said the fund was drawn to Ten63's ability to "quickly and accurately simulate trillions of potential drugs" and to "creating medicines for targets no one else can."

Company Origins, Leadership, and Academic Roots

Ten63 Therapeutics is a spinout from Duke University and the Toyota Technological Institute at Chicago (TTIC), the company said. The academic origins suggest that foundational computational methods underlying the BEYOND platform were developed in or informed by research conducted at these institutions, though the company has not publicly detailed the specific intellectual property arrangements involved.

Frenkel, who holds a Ph.D. and leads the company as CEO, has been the primary public spokesperson for Ten63. Clay Thorp, General Partner at Hatteras Venture Partners, serves as Chairman of the Board. The company's research collaboration with the University of Oxford, focused on HPV target biology and validation, represents an additional academic link, though Oxford's involvement appears to be in a collaborator capacity rather than as a source of the core AI platform technology.

Previous Funding and Partnership Activity

The company has not publicly detailed the structure or timing of its prior funding rounds. The current financing brings cumulative capital raised to more than USD 45 million, indicating that earlier rounds — likely including seed and Series A–equivalent tranches — contributed the balance. Hatteras Venture Partners, Yosemite, Morpheus Ventures, Alexandria Venture Investments, and Draper Associates are identified as existing investors who participated in prior rounds.

On the partnership front, Ten63's most visible external arrangement is the Gates Foundation–supported collaboration with the University of Oxford on HPV therapeutics. No traditional pharmaceutical out-licensing or co-development agreements have been publicly announced. The company has stated it is pursuing "select, strategic partnerships across multiple indications" alongside its internal pipeline, suggesting that partnering activity may expand as preclinical programs mature.

The AI drug discovery sector continues to draw capital, though investor scrutiny of platform companies has increased as the field matures and demands for clinical validation grow. Ten63's ability to advance its Myc and HPV programs toward investigational new drug–enabling studies will likely determine the trajectory of its next financing and partnering milestones.


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